发明名称 |
Transition metal catalyzed synthesis of 2H-indazoles |
摘要 |
The present invention relates to a process for the regioselective synthesis of compounds of the formula I, wherein R0; R1; R2; R3; R4; R5; A1; A2; A3; A4, Q and J have the meanings indicated in the claims. The present invention provides a direct transition metal catalyzed process to a wide variety of multifunctional 2H-indazoles or 2H-azaindazoles of the formula (I) from 2-halo-phenylacetylenes or (2-sulfonato)phenylacetylenes and monosubstituted hydrazines. |
申请公布号 |
US8283476(B2) |
申请公布日期 |
2012.10.09 |
申请号 |
US20090644371 |
申请日期 |
2009.12.22 |
申请人 |
HALLAND NIS;NAZARE MARC;LINDENSCHMIDT ANDREAS;ALONSO JORGE;RKYEK OMAR;URMANN MATTHIAS;SANOFI |
发明人 |
HALLAND NIS;NAZARE MARC;LINDENSCHMIDT ANDREAS;ALONSO JORGE;RKYEK OMAR;URMANN MATTHIAS |
分类号 |
C07D231/56 |
主分类号 |
C07D231/56 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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