发明名称 |
PROCESS FOR THE PREPARATION OF Y(1R), 2S -2-AMINOPROPIONIC ACID 2-Y4-(4-FLUORO-2-METHYL-1H-INDOL-5-YLOXY)-5-METHYLPYRROLOY2,1-f Y1,2,4 TRIAZIN-6-YLOXY -1-METHYLETHYL ESTER |
摘要 |
<p>The invention relates to an improved process for preparing [(1R), 2S]-2-aminopropionic acid 2-[4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-methylpyrrolo[2,1-f][1,2,4]triazin-6-yloxy]-1-methylethyl ester of the formula: Compound I has been shown to be useful for the treatment of certain types of cancer.</p> |
申请公布号 |
SI2010538(T1) |
申请公布日期 |
2013.06.28 |
申请号 |
SI20070031167T |
申请日期 |
2007.04.19 |
申请人 |
BRISTOL-MYERS SQUIBB COMAPANY |
发明人 |
CRISPINO GERARD A.;HAMEDI MOURAD;LAPORTE THOMAS L.;THORNTON JOHN E.;PESTI JAAN A.;XU ZHONGMIN;LOBBEN PAUL C.;LEAHY DAVID K.;MUSLEHIDDINOGLU JALE;LAI CHIAJEN;SPANGLER LORI ANN;DISCORDIA ROBERT P. |
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