摘要 |
Compounds of formula (I): (I) wherein Het, R3, R4, R5, R7, R8, R9, T, p, p', q, and q' are as defined in the description are pro-apoptotic agents useful in the treatment of cancers and of auto-immune and immune system diseases. |
申请人 |
VERNALIS (R&D) LIMITED;LES LABORATOIRES SERVIER |
发明人 |
DAVIDSON, JAMES EDWARD PAUL;MURRAY, JAMES BROOKE;CHEN, I-JEN;WALMSLEY, CLAIRE;DODSWORTH, MARK;MEISSNER, JOHANNES W.G.;BROUGH, PAUL;FEJES, IMRE;TATAI, JANOS;NYERGES, MIKLOS;KOTSCHY, ANDRAS;SZLAVIK, ZOLTAN;GENESTE, OLIVIER;LE TIRAN, ARNAUD;LE DIGUARHER, THIERRY;HENLIN, JEAN-MICHEL;STARCK, JEROME-BENOIT;GUILLOUZIC, ANNE-FRANCOISE;DE NANTEUIL, GUILLAUME |