发明名称 |
PRODRUG DERIVATIVES OF (E)-N-METHYL-N-((3-METHYLBENZOFURAN-2-YL)METHYL)-3-(7-OXO-5,6,7,8-TETRAHYDRO-1,8-NAPHTHYRIDIN-3-YL)ACRYLAMIDE |
摘要 |
In part, the present disclosure is directed to prodrug derivatives of (E)-N-methyl-N-((3-methylbenzofuran-2-yl)methyl)-3-(7-oxo-5,6,7,8-tetrahydro-1,8-naphthyridin-3-yl)acrylamide compounds with significant solubility and bioavailability profiles. |
申请公布号 |
SG11201408100Y(A) |
申请公布日期 |
2015.01.29 |
申请号 |
SG11201408100Y |
申请日期 |
2013.06.19 |
申请人 |
DEBIOPHARM INTERNATIONAL SA |
发明人 |
PARTRIDGE, JOHN, J.;COLUCCI, JOHN;GAREAU, YVES;THERIEN, MICHEL;ZAMBONI, ROBERT;HAFKIN, BARRY;MARFAT, ANTHONY;ZAGHDANE, HELMI |
分类号 |
C07F9/6561;A61K31/675;A61P31/04;C07F9/60 |
主分类号 |
C07F9/6561 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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