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发明名称
PROCESS FOR THE PREPARATION OF PLEUROMUTILINS
摘要
<p>본 발명은, 고순도의 산물의 대량 제조에 적합하며, 황 원자에 부착된 피페리딘 고리에서 탄소 원자가 (S)-구조 또는 (R)-구조 중 어느 하나인, 식 (I)의 14-O-[(N-(3-메틸-2-아미노-부티릴-피페리디닐)설파닐)아세틸]뮤틸린의 제조 방법, 및 14-O-[(N-(3-메틸-2-(R)-아미노-부티릴-피페리딘-3(S)-일)설파닐)아세틸]뮤틸린 염산염의 신규한 결정체 형태에 관한 것이다.</p>
申请公布号
KR101577675(B1)
申请公布日期
2015.12.15
申请号
KR20097008971
申请日期
2007.10.03
申请人
나브리바 테라퓨틱스 아게
发明人
마처 인골프;버거 안드레아스;디크리스토포로 마틴
分类号
A61K31/445;A61P31/04;C07D211/54
主分类号
A61K31/445
代理机构
代理人
主权项
地址
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