发明名称 |
QUINOXALINE-CONTAINING COMPOUNDS AS HEPATITIS C VIRUS INHIBITORS |
摘要 |
THE PRESENT INVENTION DISCLOSES COMPOUNDS OF FORMULA I AND II OR PHARMACEUTICALLY ACCEPTABLE SALTS, ESTERS, OR PRODRUGS THEREOF: WHICH INHIBIT SERINE PROTEASE ACTIVITY, PARTICULARLY THE ACTIVITY OF HEPATITIS C VIRUS (HCV) NS3-NS4A PROTEASE. CONSEQUENTLY, THE COMPOUNDS OF THE PRESENT INVENTION INTERFERE WITH THE LIFE CYCLE OF THE HEPATITIS C VIRUS AND ARE ALSO USEFUL AS ANTIVIRAL AGENTS. THE PRESENT INVENTION FURTHER RELATES TO PHARMACEUTICAL COMPOSITIONS COMPRISING THE AFOREMENTIONED COMPOUNDS FOR ADMINISTRATION TO A SUBJECT SUFFERING FROM HCV INFECTION. THE INVENTION ALSO RELATES TO METHODS OF TREATING AN HCV INFECTION IN A SUBJECT BY ADMINISTERING A PHARMACEUTICAL COMPOSITION COMPRISING THE COMPOUNDS OF THE PRESENT INVENTION. |
申请公布号 |
MY155851(A) |
申请公布日期 |
2015.12.15 |
申请号 |
MY2010PI02236 |
申请日期 |
2008.11.14 |
申请人 |
ENANTA PHARMACEUTICALS, INC. |
发明人 |
GAI, YONGHUA;OR, YAT SUN;WANG, ZHE |
分类号 |
A01N43/60 |
主分类号 |
A01N43/60 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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