发明名称 2,6,7,8 SUBSTITUTED PURINES AS HDM2 INHIBITORS
摘要 The present invention provides 2,6,7,8 Substituted Purines as described herein or a pharmaceutically acceptable salt thereof. The representative compounds are useful as inhibitors of the HDM2 protein. Also disclosed are pharmaceutical compositions comprising the above compounds and potential methods of treating cancer using the same.
申请公布号 EP2951180(A1) 申请公布日期 2015.12.09
申请号 EP20140745870 申请日期 2014.01.29
申请人 MERCK SHARP & DOHME CORP. 发明人 CAMMARANO, CAROLYN MICHELE;CHRISTOPHER, MATTHEW, P.;DINSMORE, CHRISTOPHER;DOLL, RONALD, J.;FRADERA LLINAS, FRANCESC XAVIER;LI, CHAOMIN;MACHACEK, MICHELLE;MARTINEZ, MICHELLE;NAIR, LATHA, G.;PAN, WEIDONG;REUTERSHAN, MICHAEL HALE;SHIZUKA, MANAMI;STEINHUEBEL, DIETRICH, P.;SUN, BINYUAN;THOMPSON, CHRISTOPHER FRANCIS;TROTTER, B. WESLEY;VOSS, MATTHEW ERNST;WANG, YAOLIN;YANG, LIPING;PANDA, JAGANNATH;KURISSERY, ANTHAPPAN TONY;BOGEN, STEPHANE, L.
分类号 C07D473/00;A61K31/52;A61P35/00;C07D473/16;C07D473/30;C07D473/34 主分类号 C07D473/00
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