发明名称 polimorfos de acil sulfonamidas
摘要 The application discloses novel polymorphic crystalline forms of 2-[4-Bromo-3-(3-chloro-5-cyano-phenoxy)-2-fluoro-phenyl]-N-(2-chloro-4-propionylsulfamoyl-phenyl)-acetamide, sodium salt (Ib) with improved stability and physical properties which facilitate manufacturing, handling and formulating for treatment or prophylaxis of HIV mediated diseases, AIDS or ARC, in monotherapy or in combination therapy.
申请公布号 BRPI0918526(A2) 申请公布日期 2015.12.01
申请号 BR2009PI18526 申请日期 2009.08.31
申请人 F. HOFFMANN-LA ROCHE AG 发明人 FEI PANG;JAMES PRENTICE DAVIDSON;MAGARET WONG;MICHAEL MARTIN
分类号 C07C303/44;C07C311/51 主分类号 C07C303/44
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