发明名称 |
PROCESSES OF MAKING AND CRYSTALLINE FORMS OF A MDM2 INHIBITOR |
摘要 |
The present invention provides processes for making 2-((3R,5R,6S)-5-(3-chlorophenyl)-6-(4-chlorophenyl)-1-((S)-1-(isopropylsulfonyl)-3-methylbutan-2-yl)-3-methyl-2-oxopiperidin-3-yl)acetic acid as well as intermediates and processes for making the intermediates. Also provided are crystalline forms of the compound and the intermediates. |
申请公布号 |
AP201508891(D0) |
申请公布日期 |
2015.11.30 |
申请号 |
AP20150008891 |
申请日期 |
2014.06.09 |
申请人 |
AMGEN INC |
发明人 |
WORTMAN SARAH;WIEDEMANN SEAN;VOUNATSOS FILISATY |
分类号 |
C07D498/04;A61K31/45;C07C309/04;C07D211/76 |
主分类号 |
C07D498/04 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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