发明名称 PROCESS FOR MAKING MODULATORS OF CYSTIC FIBROSIS TRANSMEMBRANE CONDUCTANCE REGULATOR
摘要 The invention provides a process for the preparation of a compound of Formula 1; comprising coupling a carboxylic acid of Formula 2; with an aniline of Formula 2; in the presence of a coupling agent.
申请公布号 HRP20151137(T1) 申请公布日期 2015.11.20
申请号 HR2015P001137T 申请日期 2015.10.27
申请人 VERTEX PHARMACEUTICALS INCORPORATED 发明人 DEMATTEI, JOHN;LOOKER, ADAM R.;NEUBERT-LANGILLE, BOBBIANNA;TRUDEAU, MARTIN;ROEPER, STEFANIE;RYAN, MICHAEL P.;YAP, DAHRIKA MILFRED LAO;KRUEGER, BRIAN R.;GROOTENHUIS, PETER D. J.;VAN GOOR, FREDERICK F.;BOTFIELD, MARTYN C.;ZLOKARNIK, GREGOR
分类号 C07D215/233 主分类号 C07D215/233
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