发明名称 POLYMORPHIC AND AMORPHOUS FORMS OF CORTISOL 17-ALPHA-BENZOATE AND METHODS FOR THE PREPARATION AND USE THEREOF
摘要 <p>Provided herein are multiple solid forms of a defined steroid-like compound, and methods for the preparation and use thereof. In one aspect, there is provided a crystalline form of said steroid-like compound, and methods for the preparation and use thereof. In another aspect, there is provided a substantially amorphous form of said steroid-like compound, and methods for the preparation and use thereof. In yet another aspect, there are provided compositions containing compounds according to the present invention. In certain aspects, such compositions are suitable for delivery of active agents according to the present invention to a subject in need thereof. In another aspect of the invention, there are provided methods for the treatment of a variety of indications, including glaucoma, ocular hypertension, and the like. In still another aspect of the present invention, there are provided kits containing compounds according to the present invention and/or compositions containing same.</p>
申请公布号 WO2015089471(A3) 申请公布日期 2015.11.19
申请号 WO2014US70147 申请日期 2014.12.12
申请人 ALLERGAN, INC. 发明人 FENG, SHAOXIN;SMITH, SCOTT W.;LAMBERT, OLIVIER M.G.;BUTTAR, SUZANNE
分类号 C07J5/00;A61K31/573;A61P27/06 主分类号 C07J5/00
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