发明名称 |
CRYSTALLINE (S)-ISOPROPYL 2-(((S)-(((2R,3R,4R,5R)-5-(2,4-DIOXO-3,4-DIHYDROPYRIMIDIN-1-(2H)-YL)-4-FLUORO-3-HYDROXY-4-METHYLTETRAHYDROFURAN-2-YL)METHOXY)(PHENOXY)PHOSPHORYL)AMINO)PROPANOATE |
摘要 |
<p>Disclosed herein are phosphorus-containing actives, their use as actives for treating diseases, and a stereoselective process for preparing the same. Also disclosed herein are useful synthetic intermediates and processes for preparing the same.</p> |
申请公布号 |
PT2552930(E) |
申请公布日期 |
2015.11.17 |
申请号 |
PT20110714465T |
申请日期 |
2011.03.31 |
申请人 |
GILEAD PHARMASSET LLC |
发明人 |
BYOUNG-KWON CHUN;MICHAEL JOSEPH SOFIA;BRUCE S. ROSS;GANAPATI REDDY PAMULAPATI;SUGUNA RACHAKONDA;HAI-REN ZHANG;PEIYUAN WANG |
分类号 |
C07H19/10;A61K31/7072;A61P31/14 |
主分类号 |
C07H19/10 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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