发明名称 |
A PROCESS FOR PREPARING [1S- ]1-ALPHA, 2-ALPHA, 3-BETA (1S*, 2R*) 5-BETA] ]-3- [7- [2- (3, 4-DIF LUOROPHENYL) -CYCLOPROPYLAMINO]- 5- (PROPYLTHIO) -3H-1, 2, 3-TRIAZOLO [4, 5-D]PYRIMIDIN-3-YL]-5- (2- HYDROXYETHOXY) CYCLOPENTANE-1, 2-DIOL AND TO ITS INTERMEDIATES |
摘要 |
The present invention is directed to a process for preparing [1S-[1alpha,2alpha,3beta(1S*,2R*),5beta]]-3-[7-[2-(3,4-difluorophenyl)-cyclopropylamino]-5-(propylthio)-3H-1,2,3-triazolo[4,5-d]pyrimidin-3-yl]-5-(2-hydroxyethoxy)cyclopentane-1,2-diol and to intermediates useful in the process. |
申请公布号 |
EP2340252(B1) |
申请公布日期 |
2015.11.11 |
申请号 |
EP20090813307 |
申请日期 |
2009.09.08 |
申请人 |
ASTRAZENECA AB |
发明人 |
AUFDENBLATTEN, RHONY;BOHLIN, MARTIN, HANS;HELLSTRÖM, HELENA;JOHANSSON, PETER, W;LARSSON, ULF, G;RECKNAGEL, MIKAELA;WEISS, URSULA, HEIRESS OF WEISS ANDREAS (DECEASED) |
分类号 |
C07D487/04;C07D317/44;C07D405/04;C07D405/12 |
主分类号 |
C07D487/04 |
代理机构 |
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代理人 |
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