| 发明名称 |
PROCESSES AND INTERMEDIATES FOR THE PREPARATION OF A PDE10 INHIBITOR |
| 摘要 |
The present invention is directed to an improved process for the preparation of compounds of Formula (II) and Formula (III), which are useful in the inhibition of PDE10. In particular, the present invention is directed to an improved process for the preparation of 1-(5-(4-chloro-3,5-dimethoxyphenyl)furan-2-yl)-2-ethoxy-2-(4-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl)ethanone, which is useful in the inhibition of PDE10. |
| 申请公布号 |
WO2015167969(A1) |
申请公布日期 |
2015.11.05 |
| 申请号 |
WO2015US27647 |
申请日期 |
2015.04.24 |
| 申请人 |
OMEROS CORPORATION |
发明人 |
CUTSHALL, NEIL S.;GAGE, JENNIFER LYNN;LITTLE, THOMAS L.;LUKE, WAYNE DOUGLAS;BROT, ELISABETH C.A.;JONAS, MARCO;MCDERMOTT, MICHAEL JAMES;REINEKE, KARL E. |
| 分类号 |
C07D417/10 |
主分类号 |
C07D417/10 |
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