主权项 |
1. A compound selected from the following group:No.Name“A1”2-p-tolyl-3H-pyrrolo[2,1-f][1,2,4]triazin-4-one“A2”4-(4-oxo-3,4-dihydro-pyrrolo[2,1-f][1,2,4]triazin-2-yl)-benzoicacid methyl ester“A3”2-(4-tert-butyl-phenyl)-3H-pyrrolo[2,1-f][1,2,4]triazin-4-one“A4”2-(1-acetyl-piperidin-4-yl)-3H-pyrrolo[2,1-f][1,2,4]triazin-4-one“A5”2-[4-(1-hydroxy-1-methyl-ethyl)-phenyl]-3H-pyrrolo-[2,1-f][1,2,4]triazin-4-one“A6”2-(4-bromo-phenyl)-3H-pyrrolo[2,1-f][1,2,4]triazin-4-one“A7”2-[4-(1-methyl-1H-pyrazol-4-yl)-phenyl]-3H-pyrrolo-[2,1-f][1,2,4]triazin-4-one“A8”2-(4-pyrrolidin-l-ylphenyl)-3H-pyrrolo[2,1-f][1,2,4]triazin-4-one“A9”2-cyclohexyl-3H-pyrrolo[2,1-f][1,2,4]triazin-4-one“A10”2-(1-tert-butylpyrazol-4-yl)-3H-pyrrolo[2,1-f][1,2,4]triazin-4-one“A11”2-[4-(1-hydroxy-1-methyl-ethyl)phenyl]-6-methyl-3H-pyrrolo [2,1-f][1,2,4]triazin-4-one“A12”6-fluoro-2-[4-(1-hydroxy-1-methyl-ethyl)phenyl]-3H-pyrrolo [2,1-f][1,2,4]triazin-4-one“A13”6-methyl-2-[4-(1-methylpyrazol-4-yl)phenyl]-3H-pyrrolo-[2,1-f][1,2,4]triazin-4-one“A14”2-[4-(1-ethyl-1-hydroxy-propyl)-phenyl]-3H-pyrrolo[2,1-f][1,2,4]triazin-4-one“A15”2-{4-[1-(2-hydroxy-ethoxy)-1-methyl-ethyl]-phenyl}-3H-pyrrolo[2,1-f][1,2,4]triazin-4-one“A16”2-[4-(1-amino-1-methyl-ethyl)-phenyl]-3H-pyrrolo[2,1-f][1,2,4]-triazin-4-one“A17”6-[4-(1-hydroxy-1-methyl-ethyl)-phenyl]-2-methyl-5H-1,5,7,7a-tetraaza-inden-4-one“A18”6-chloro-2-[4-(1-hydroxy-1-methyl-ethyl)-phenyl]-3H-pyrrolo [2,1-f][1,2,4]triazin-4-one“A19”2-[4-(1-hydroxy-1-methyl-ethyl)-phenyl]-7-methyl-3H-pyrrolo[2,1-f][1,2,4]triazin-4-one“A20”2-[4-(1-hydroxy-1-methyl-ethyl)-phenyl]-7-trifluoromethyl-3H-pyrrolo[2,1-f][1,2,4]triazin-4-one“A21”2-[4-(1-hydroxy-cyclopentyl)-phenyl]-3H-pyrrolo[2,1-f][1,2,4]-triazin-4-one and pharmaceutically acceptable solvates, salts, tautomers and stereoisomers thereof, including mixtures thereof in all ratios. |