发明名称 |
1H-PYRROLO[2,3-c]PYRIDIN-7(6H)-ONES AND PYRAZOLO[3,4-c]PYRIDIN-7(6H)-ONES AS INHIBITORS OF BET PROTEINS |
摘要 |
The present invention relates to substituted pyrrolopyridinones and substituted pyrazolopyridinones which are inhibitors of BET proteins such as BRD2, BRD3, BRD4, and BRD-t and are useful in the treatment of diseases such as cancer. |
申请公布号 |
WO2015164480(A1) |
申请公布日期 |
2015.10.29 |
申请号 |
WO2015US27047 |
申请日期 |
2015.04.22 |
申请人 |
INCYTE CORPORATION |
发明人 |
COMBS, ANDREW, P.;MADUSKUIE, THOMAS, P., JR.;FALAHATPISHEH, NIKOO |
分类号 |
C07D471/04;A61K31/437;A61P9/10;A61P11/06;A61P25/24;A61P25/28;A61P31/00;A61P33/00;A61P35/00;A61P37/00 |
主分类号 |
C07D471/04 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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