发明名称 Aminopyrimidines as Syk inhibitors
摘要 <p>AMINOPYRIMIDINES AS SYK INHIBITORS Abstract The present invention provides novel pyrimidine amines of formula (I) which are potent inhibitors of spleen tyrosine kinase, and are useful in the treatment and prevention of diseases mediated by said enzyme, such as asthma, COPD and rheumatoid arthritis.</p>
申请公布号 AU2014200138(A8) 申请公布日期 2015.10.29
申请号 AU20140200138 申请日期 2014.01.10
申请人 MERCK CANADA INC.;MERCK SHARP & DOHME CORP. 发明人 ALTMAN, MICHAEL D.;ANDRESEN, BRIAN M.;ARRINGTON, KENNETH L.;CHILDERS, KALEEN KONRAD;DI FRANCESCO, MARIA EMILIA;DONOFRIO, ANTHONY;ELLIS, JOHN MICHAEL;FISCHER, CHRISTIAN;GUERIN, DAVID JOSEPH;HAIDLE, ANDREW M.;KATTAR, SOLOMON;KNOWLES, SANDRA LEE;LI, CHAOMIN;LIM, JONGWON;MACHACEK, MICHELLE R.;NORTHRUP, ALAN B.;O'BOYLE, BRENDAN M.;OTTE, RYAN D.;PETROCCHI, ALESSIA;REUTERSHAN, MICHAEL H.;ROMEO, ERIC;SIU, TONY;TAOKA, BRANDON M.;TROTTER, B. WESLEY;ZHOU, HUA;BURCH, JASON;COTE, BERNARD;DUPONT-GAUDET, KRISTINA;FOURNIER, JEAN-FRANCOIS;GAUTHIER, JACQUES YVES;GUAY, DANIEL;ROBICHAUD, JOEL S.;GRIMM, JONATHAN;MADDESS, MATTHEW L.;SCHELL, ADAM J.;SPENCER, KERRIE B.;WOO, HYUN CHONG;BHAT, SATHESH
分类号 C07D417/12;A61K31/497;A61P11/00;A61P11/06;A61P29/00;A61P35/00;C07D417/14 主分类号 C07D417/12
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