发明名称 1H-pyrrolo(2,3-c)pyridin-7(6H)-ones and pyrazolo(3,4-C)pyridin-7(6H)-ones as inhibitors of BET proteins
摘要 The present invention relates to substituted pyrrolopyridinones and substituted pyrazolopyridinones which are inhibitors of BET proteins such as BRD2, BRD3, BRD4, and BRD-t and are useful in the treatment of diseases such as cancer.
申请公布号 AU2015249810(A1) 申请公布日期 2015.10.29
申请号 AU20150249810 申请日期 2015.04.22
申请人 Incyte Corporation 发明人 Combs, Andrew P.;Maduskuie Jr., Thomas P.;Falahatpisheh, Nikoo
分类号 C07D471/04;A61K31/437;A61P9/10;A61P11/06;A61P25/24;A61P25/28;A61P31/00;A61P33/00;A61P35/00;A61P37/00 主分类号 C07D471/04
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