发明名称 CRYSTAL FORM OF COMPOUND USED AS MINERALOCORTICOID RECEPTOR ANTAGONIST AND PREPARATION METHOD THEREFOR
摘要 The present invention belongs to the technical field of medicines, and relates to a crystal form of a compound used as a mineralocorticoid receptor antagonist and a preparation method therefor, and in particular, to a method for preparing a compound 2-chloro-4-[(3S,3aR)-3-cyclopentyl-7-(4-hydroxypiperidin-1-carbonyl)-3,3a,4,5-tetrahydro-2H -pyrazolo[3,4-f]quinolin-2-yl]benzonitrile of formula (1); a crystal form thereof, a preparation method for the crystal form, and the use of the crystal form in the preparation of drugs for the treatment and/or prevention of renal injury or cardiovascular diseases.
申请公布号 EP2937348(A1) 申请公布日期 2015.10.28
申请号 EP20130864994 申请日期 2013.12.23
申请人 KBP BIOSCIENCES CO., LTD. 发明人 JIANG, CHEN;WANG, AICHEN;ZHANG, DEDONG
分类号 C07D471/04;A61K31/4745;A61P5/40;A61P7/00;A61P9/00;A61P9/04;A61P9/06;A61P9/10;A61P9/12;A61P13/12;A61P25/00;A61P29/00 主分类号 C07D471/04
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