发明名称 |
CRYSTALLINE FORMS AND PROCESSES FOR THE PREPARATION OF PHENYL-PYRAZOLES USEFUL AS MODULATORS OF THE 5-HT2A SEROTONIN RECEPTOR 5-HT2A |
摘要 |
<p>The present invention relates to processes for preparing phenyl-pyrazoles of Formula (I) and salts and pharmaceutical compositions thereof, useful as modulators of 5-HT 2A serotonin receptor activity. The present invention also relates to intermediates used in the processes, and their preparation. The present invention also relates to crystalline forms of 5-HT 2A serotonin receptor modulators, compositions thereof and methods of using the same.</p> |
申请公布号 |
HK1121453(A1) |
申请公布日期 |
2015.10.23 |
申请号 |
HK20090101461 |
申请日期 |
2009.02.17 |
申请人 |
ARENA PHARMACEUTICALS INC. |
发明人 |
TAWFIK GHARBAOUI;DIPANJAN SENGUPTA;ASHWIN M. KRISHNAN;NAINESH SHAH;MARK MACIAS;RYAN M. HART;EDWARD A. LALLY;JONATHAN J DUFFIELD |
分类号 |
C07D;A61K;A61P |
主分类号 |
C07D |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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