| 主权项 |
1. A compound of Formula II: wherein (I) G is and, Cy is aryl or heteroaryl, said aryl or heteroaryl being optionally substituted with one or more R1 substituents, or, (II) G is and, Cy is
a) a six-membered carbocyclic aromatic ring substituted with one or more R1 substituents;b) a six-membered carbocyclic aromatic ring fused to a saturated or aromatic five-membered carbocyclic ring, wherein said fused rings are optionally substituted with one or more R1 substituents;c) a six-membered carbocyclic aromatic ring fused to a saturated, unsaturated, or aromatic six-membered carbocyclic ring, wherein said fused rings are optionally substituted with one or more R1 substituents; or,d) heteroaryl that is optionally substituted with one or more R1 substituents; R1 is
halogen,NO2,CN,C1-C6 alkyl,NR5R6,COR4,C(O)OR4,S(O)2R4,(CONR5R6)1-3, orS(O)2NR5R6, wherein alkyl is optionally substituted with one or more R7 substituents; wherein when G is (1), R2 is
H,halogen,NO2,CN,C1-C6 alkyl,NR5R6,COR4;C(O)OR4;S(O)2R4;(CONR5R6)1-3, orS(O)2NR5R6, wherein alkyl is optionally substituted with one or more R7 substituents; wherein when G is (2) or (4), R2 and R3 are each independently
H,halogen,NO2,CN,C1-C6 alkyl,NR5R6,COR4;C(O)OR4;S(O)2R4;(CONR5R6)1-3, orS(O)2NR5R6, or, R2 and R3 together with the carbon atoms to which they are attached form a benzene ring, wherein alkyl is optionally substituted with one or more R7 substituents; wherein when G is (3), R2 is
H,halogen,CN,C1-C6 alkyl,COR4;C(O)OR4;S(O)2R4;(CONR5R6)1-3, orS(O)2NR5R6, wherein alkyl is optionally substituted with one or more R7 substituents, and, R3 is
H,halogen,NO2,CN,C1-C6 alkyl,NR5R6,COR4;C(O)OR4;S(O)2R4;(CONR5R6)1-3, orS(O)2NR5R6, wherein alkyl is optionally substituted with one or more R7 substituents; R4 is
1) C1-C6 alkyl,2) aryl, or3) heteroaryl, R5 and R6 are independently
1) H, or2) C1-C6 alkyl, or, R5 and R6 together with the nitrogen atom to which they are bonded form a five or six membered heterocyclic ring; wherein alkyl is optionally substituted with one or more R7 substituents; and, R7 is
1) halogen,2) NO2,3) CN,4) C1-C6 alkyl,5) haloalkyl,6) OR4,7) NH2, N(C1-C6 alkyl)2 or NH(C1-C6 alkyl),8) SR4,9) COR4,10) C(O)OR4,11) S(O)2R4,12) CONH2, CON (C1-C6 alkyl)2 or CONH(C1-C6 alkyl), or13) S(O)2NH2 S(O)2N(C1-C6alkyl)2 or S(O)NH (C1-C6 alkyl). |
