发明名称 Cyklisk pyrimidin-4-carboxamider, som CCR2-receptor-antagonister til behandling af inflammation, astma og COPD
摘要 <p>The present invention relates to a process for the production of novel antagonists for CCR2 (CC chemokine receptor 2) of formula (I) from 6-Chloro-pyrimidine-methanone intermediates. Formula (I): Specifically claimed 6-chloropyrimidine-methanone intermediates are:</p>
申请公布号 DK2379525(T3) 申请公布日期 2015.10.19
申请号 DK20090775212T 申请日期 2009.12.17
申请人 BOEHRINGER INGELHEIM INTERNATIONAL GMBH 发明人 EBEL, HEINER;FRATTINI, SARA;GIOVANNINI, RICCARDO;HOENKE, CHRISTOPH;TRIESELMANN, THOMAS;TIELMANN, PATRICK;SCHEUERER, STEFAN;HOBBIE, SILKE (MARIE KATRIN);BUETTNER, FRANK
分类号 C07D405/14;A61K31/506;A61K31/5377;A61K31/55;A61K31/551;A61K31/553;C07D401/06;C07D401/14;C07D403/06;C07D403/14;C07D407/14;C07D413/14;C07D417/14;C07D451/02;C07D471/04;C07D471/10;C07D491/052;C07D498/10 主分类号 C07D405/14
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