发明名称 |
PROCESSES FOR PREPARATION OF S1P1 RECEPTOR MODULATORS AND CRYSTALLINE FORMS THEREOF |
摘要 |
<p>PROBLEM TO BE SOLVED: To provide processes for preparation of S1P1 receptor modulators and crystalline forms thereof.SOLUTION: The present invention relates to salts, processes, and process intermediates useful in the preparation of (R)-2-(9-chloro -7-(4-isopropoxy-3-(trifluoromethyl)benzyloxy)-2,3-dihydro-1H-pyrrolo[1,2-a]indole-1-yl)acetic acid of formula (Ia), and salts and crystalline forms thereof.</p> |
申请公布号 |
JP2015180706(A) |
申请公布日期 |
2015.10.15 |
申请号 |
JP20150142650 |
申请日期 |
2015.07.17 |
申请人 |
ARENA PHARMACEUTICALS INC |
发明人 |
JONES ROBERT M;DANIEL J BUZARD;TAWFIK GHARBAOUI;BENJAMIN R JOHNSON;MICHELLE KASEM;THOMAS O SCHRADER;SCOTT STIRN |
分类号 |
C07D487/04;A61K31/407;A61P1/04;A61P1/16;A61P3/10;A61P5/00;A61P9/10;A61P13/12;A61P17/06;A61P17/10;A61P21/00;A61P25/00;A61P29/00;A61P37/06;A61P43/00 |
主分类号 |
C07D487/04 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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