发明名称 SYNTHESIS OF VORTIOXETINE VIA (2,4-DIMETHYLPHENYL)(2-IODOPHENYL)SULFANE INTERMEDIATE
摘要 The present invention provides a new synthetic process for the production of 1 -(2-((2,4-dimethylphenyl)thio)phenyl)piperazine (vortioxetine), a drug for the treatment of depression and anxiety, which is conducted via (2,4-dimethylphenyl)(2-iodophenyl)sulfane intermediate.
申请公布号 WO2015155153(A1) 申请公布日期 2015.10.15
申请号 WO2015EP57444 申请日期 2015.04.07
申请人 LEK PHARMACEUTICALS D.D. 发明人 ZUPANCIC, BORUT
分类号 C07D295/096;A61K31/495;A61P25/24 主分类号 C07D295/096
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