发明名称 AMINO ACID PRECURSOR, AMINO ACID, AND PRODUCTION METHOD FOR AMINO ACID, AND PET DIAGNOSTIC TRACER USING AMINO ACID
摘要 Disclosed is an amino acid that can be prevented from being incorporated into normal cells and selectively incorporated into tumor cells, even when used in a PET diagnostic tracer. Also disclosed are an amino acid precursor, a production method for the amino acid, and a PET diagnostic tracer that uses the amino acid. The amino acid of the present invention is represented by formula (II). The amino acid of the present invention is, for example, useful as a PET diagnostic tracer or as a building block for a pharmaceutical intermediate.
申请公布号 WO2015152128(A1) 申请公布日期 2015.10.08
申请号 WO2015JP59862 申请日期 2015.03.30
申请人 NAGASE & CO., LTD.;RIKEN 发明人 YAMAMOTO, KENICHIRO;KODAMA, KAZUYA;SASANO, YUMI;HUME, WILLIAM EWAN;YASHIO, KEIJI;NOZAKI, SATOSHI
分类号 C07C229/36;A61K51/00;C07B57/00;C07B59/00 主分类号 C07C229/36
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