发明名称 |
Compuestos derivados de heterociclos nitrogenados, moduladores de quinasas; metodo de preparacion; compuesto iintermediario; composicion farmaceutica; y un metodo para tratar un sujeto que posee una enferemedad o condicion como cancer, aml, tumores estromales gastrointestinales o mastocitosis. |
摘要 |
Compounds active on c-kit protein kinases or mutant c-kit protein kinases having any mutations are described, as well as methods of making and using such compounds to treat diseases and conditions associated with aberrant activity of the c-kit protein kinases and/or mutant c-kit protein kinases. |
申请公布号 |
CL2015001785(A1) |
申请公布日期 |
2015.10.02 |
申请号 |
CL20150001785 |
申请日期 |
2015.06.19 |
申请人 |
PLEXXIKON, INC. |
发明人 |
IBRAHIM PRABHA N.;SPEVAK WAYNE;EWING TODD;ZHANG YING;WU. GUOXIAN;CHAN KATRINA;LIN JACK;NESPI MARIKA |
分类号 |
C07D401/12;A61K31/437;A61P35/00;C07D403/12;C07D471/04;C07D487/04;C07D513/04 |
主分类号 |
C07D401/12 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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