发明名称 |
SULFONAMIDO-ALKYL-CARBOXAMIDO-METHYL-PIPERIDINE AND MORPHOLINE DERIVATIVES |
摘要 |
THE NOVEL SULPHONAMIDOCARBOXAMIDES OF THE FORMULA(FORMULA 1)WHEREIN A, M, Q, X AND Y HAVE THE SIGNIFICANCE GIVEN IN THE DESCRIPTION, AS WELL AS HYDRATES OR SOLVATES THEREOF INHIBIT THROMBIN-INDUCED BLOOD PLATELET AGGREGATION AND CLOTTING OF FIBRINOGEN IN PLASMA. THEY ARE MANUFACTURED BY AMIDINATION OF A CYCLIC AMINO GROUP STANDING FOR GROUPING X OR BY C(O)N(Q) AMIDE FORMATION.
|
申请公布号 |
MY131303(A) |
申请公布日期 |
2007.08.30 |
申请号 |
MYPI9300383 |
申请日期 |
1993.03.03 |
申请人 |
F. HOFFMANN-LA ROCHE AG |
发明人 |
JEAN ACKERMANN;DAVID BANNER;KLAUS GUBERNATOR;KURT HILPERT;GERARD SCHMID |
分类号 |
A61K31/445;C07D211/26;A61K;A61K31/155;A61K31/18;A61K31/33;A61K31/435;A61K31/4427;A61K31/452;A61K31/47;A61K31/535;A61K31/5375;A61K31/63;A61K31/675;A61K38/00;A61P7/02;C07C231/00;C07C237/16;C07C277/00;C07C279/16;C07C279/18;C07C279/20;C07C311/00;C07C311/19;C07D;C07D211/18;C07D211/28;C07D211/36;C07D211/56;C07D265/06;C07D265/28;C07D265/30;C07D295/00;C07D401/12;C07D401/14;C07D413/12;C07F9/59;C07K5/06;C07K5/068;C07K5/072;C07K5/078 |
主分类号 |
A61K31/445 |
代理机构 |
|
代理人 |
|
主权项 |
|
地址 |
|