ENZYMATIC RESOLUTION OF ENDO-BICYCLO(2.2.1)HEPTAN-2-O1 AND DERIVED PHARMACEUTICAL AGENTS

摘要

Process for the pancreatic lipase mediated transesterification method for the optical resolution of endo-norborneol; derived optically active 5-(3-(exo-bicyclo[2.2.1]hept-2-yloxy)-4-methoxyphenyl)-3,4,5,6-tetrahy dropyrimid in-2(1H)-ones; and stepwise process and intermediates therefor.