发明名称 PROCESS FOR PRODUCING PIPECOLIC-2-ACID-2 ',6'-XYLIDIDE USEFUL AS AN INTERMEDIATE FOR THE PREPARATION OF LOCAL ANESTHETICS
摘要 <p>The present invention relates to an improved process for the preparation of pipecolic-2- acid-2',6'-xylidide or derivative thereof wherein it comprises hydrogenation of picolinic-2-acid-2',6'-xylidide in the presence of a Raney-nickel as a catalyst.</p>
申请公布号 WO2009089842(A1) 申请公布日期 2009.07.23
申请号 WO2008EP00237 申请日期 2008.01.15
申请人 PHARMATHEN S.A.;SONI, ROHIT, RAVIKANT;KOFTIS, THEOCHARIS;GEORGOPOULOU, IONNA;KARAGIANNIDOU, EVRYKLEIA 发明人 SONI, ROHIT, RAVIKANT;KOFTIS, THEOCHARIS;GEORGOPOULOU, IONNA;KARAGIANNIDOU, EVRYKLEIA
分类号 C07D211/60 主分类号 C07D211/60
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