发明名称 FUSED HETEROCYCLIC DERIVATIVES AND METHODS OF USE
摘要 <p>Selected compounds are effective for prophylaxis and treatment of diseases, such as HGF mediated diseases. The invention encompasses novel compounds, analogs, prodrugs and pharmaceutically acceptable salts thereof, pharmaceutical compositions and methods for prophylaxis and treatment of diseases and other maladies or conditions involving, cancer and the like. The subject invention also relates to processes for making such compounds as well as to intermediates useful in such processes.</p>
申请公布号 WO2009091374(A2) 申请公布日期 2009.07.23
申请号 WO2008US11724 申请日期 2008.10.14
申请人 AMGEN INC.;ALBRECHT, BRIAN K.;BAUER, DAVID;BELLON, STEVEN;BODE, CHRISTIANE M.;BOOKER, SHON;BOEZIO, ALESSANDRO;CHOQUETTE, DEBORAH;D'AMICO, ERIN;HARMANGE, JEAN-CHRISTOPHE;HIRAI, SATOKO;HUNGATE, RANDALL W.;KIM, TAE-SEONG;LEWIS, RICHARD T.;LIU, LONGBIN;LOHMAN, JULIA;NORMAN, MARK H.;POTASHMAN, MICHELLE;SIEGMUND, AARON C.;SPRINGER, STEPHANIE;STEC, MARKIAN;XI, NING;YANG, KEVIN;PETERSON, EMILY, A.;ROMERO, KARINA;COPELAND, KATRINA, W. 发明人 ALBRECHT, BRIAN K.;BAUER, DAVID;BELLON, STEVEN;BODE, CHRISTIANE M.;BOOKER, SHON;BOEZIO, ALESSANDRO;CHOQUETTE, DEBORAH;D'AMICO, ERIN;HARMANGE, JEAN-CHRISTOPHE;HIRAI, SATOKO;HUNGATE, RANDALL W.;KIM, TAE-SEONG;LEWIS, RICHARD T.;LIU, LONGBIN;LOHMAN, JULIA;NORMAN, MARK H.;POTASHMAN, MICHELLE;SIEGMUND, AARON C.;SPRINGER, STEPHANIE;STEC, MARKIAN;XI, NING;YANG, KEVIN;PETERSON, EMILY, A.;ROMERO, KARINA;COPELAND, KATRINA, W.
分类号 C07D471/04;A61K31/4355;C07D487/04;C07D493/04;C07D495/04;C07D498/04 主分类号 C07D471/04
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