发明名称 BICYCLIC HETEROCYCLIC COMPOUNDS AS PROTEIN TYROSINE KINASE INHIBITORS
摘要 The invention relates to new bicyclic heterocyclic derivative compounds of formula (I): wherein R1, q, A, B, X1, X2, X3, X4, X5 and R2 are as defined herein, to pharmaceutical compositions comprising said compounds and to the use of said compounds in the treatment of diseases, e.g. cancer.
申请公布号 WO2009047522(A1) 申请公布日期 2009.04.16
申请号 WO2008GB03439 申请日期 2008.10.10
申请人 ASTEX THERAPEUTICS LIMITED;SAXTY, GORDON;BERDINI, VALERIO;MURRAY, CHRISTOPHER, WILLIAM;GRIFFITHS-JONES, CHARLOTTE, MARY;VICKERSTAFFE, EMMA;BESONG, GILBERT, EBAI 发明人 SAXTY, GORDON;BERDINI, VALERIO;MURRAY, CHRISTOPHER, WILLIAM;GRIFFITHS-JONES, CHARLOTTE, MARY;VICKERSTAFFE, EMMA;BESONG, GILBERT, EBAI
分类号 C07D471/04;A61K31/437;A61P35/00;C07D487/04 主分类号 C07D471/04
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