发明名称 BENZOCYCLOHEPTENE DERIVATIVES AS ESTROGENS HAVING SELECTIVE ACTIVITY
摘要 The present invention describes non-steroidal compounds of the general formula (I) in which A is in which X1 means one or more groups on the phenyl ring and represents independently of one another a halogen, OH, (C1-C4)alkyl, (C1-C4)alkyl-O, (C3-C6)cycloalkyl-O, (C1-C14)acyl-O, (C1-C4)alkenyl, (C1-C4)alkynyl, perfluoro(C1-C4)alkyl radical, -CHO or CN, and X2 means one or more groups on the phenyl ring and represents independently of one another an H, halogen, OH, (C1-C4)alkyl, (C1-C4)alkyl-O, (C1-C4)alkenyl, (C1-C4)alkynyl, perfluoro-(C1-C4)alkyl radical, -CHO or CN, as Estrogens.
申请公布号 US2009099250(A1) 申请公布日期 2009.04.16
申请号 US20080249056 申请日期 2008.10.10
申请人 WYRWA RALF;PETERS OLAF;BOHLMANN ROLF;DROESCHER PETER;PRELLE KATJA;FRITZEMEIER KARL HEINRICH;MUHN HANS PETER 发明人 WYRWA RALF;PETERS OLAF;BOHLMANN ROLF;DROESCHER PETER;PRELLE KATJA;FRITZEMEIER KARL HEINRICH;MUHN HANS PETER
分类号 A61K31/381;A61K31/05;A61K31/122;A61P5/00;C07C39/17;C07C49/747;C07D333/16 主分类号 A61K31/381
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