发明名称 |
PROCESS AND INTERMEDIATES TO A TETRAHYDRO-[1,8]-NAPHTHYRIDINE |
摘要 |
A novel process is provided for the preparation of 3-(5,6,7,8-tetrahydro-[1,8]-naphthyridin-2-yl)-propylamine which is useful in the synthesis of .alpha.v integrin receptor antagonists. Also provided are useful intermediates obtained from the process.
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申请公布号 |
CA2391013(C) |
申请公布日期 |
2010.09.21 |
申请号 |
CA20002391013 |
申请日期 |
2000.11.20 |
申请人 |
MERCK & CO., INC. |
发明人 |
RIVERA, NELO;XIAO, YI;YASUDA, NOBUYOSHI |
分类号 |
C07D471/04;C07F9/40 |
主分类号 |
C07D471/04 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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