发明名称 FLUOROBORON COMPOUND, AMINOMETHYLATING AGENT FOR AROMATIC RING MADE OF THE SAME, AND PRODUCTION METHOD OF COMPOUND CONTAINING AMINOMETHYL AROMATIC RING USING AMINOMETHYLATING AGENT
摘要 A production method of a compound containing a primary, secondary, or tertiary aminomethyl aromatic ring of the present invention includes: using a fluoroboron compound or a dimer thereof, or solvates thereof, which are represented by a formula (I): Ra(Rb)N—CH2—BF3M  (I) as an aminomethylating agent for an aromatic ring; and reacting the aminomethylating agent with an aromatic ring-containing compound, which can react with the aminomethylating agent, under the presence of a metal catalyst such as a palladium compound so as to perform the direct aminomethylation of the aromatic ring.
申请公布号 US2012010403(A1) 申请公布日期 2012.01.12
申请号 US201113238571 申请日期 2011.09.21
申请人 TANAKA KEIGO 发明人 TANAKA KEIGO
分类号 C07F5/02;C07C209/66;C07C213/02;C07C231/10;C07C269/00;C07D209/48;C07D295/023 主分类号 C07F5/02
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