发明名称 PEPTIDOMIMETIC MACROCYCLES
摘要 The present invention provides novel peptidomimetic macrocycles and methods of using such macrocycles for the treatment of disease.
申请公布号 US2014378390(A1) 申请公布日期 2014.12.25
申请号 US201414460848 申请日期 2014.08.15
申请人 AILERON THERAPEUTICS, INC. 发明人 GUERLAVAIS Vincent;KAWAHATA Noriyuki
分类号 C07K7/64 主分类号 C07K7/64
代理机构 代理人
主权项 1. A peptidomimetic macrocycle comprising an amino acid sequence which is at least 60% identical to the amino acid sequence of: SEQ ID NO. 254, SEQ ID NO. 289, SEQ ID NO. 290, SEQ ID NO. 374, SEQ ID NO. 375, SEQ ID NO. 507, SEQ ID NO. 533, SEQ ID NO. 587, SEQ ID NO. 605, SEQ ID NO. 624, SEQ ID NO. 642, SEQ ID NO. 699, SEQ ID NO. 702, SEQ ID NO. 703, SEQ ID NO. 704, SEQ ID NO. 714, SEQ ID NO. 734, or SEQ ID NO.
地址 Cambridge MA US