发明名称 |
THIA-TRIAZA-CYCLOPENTAZULENES AS PI3-KINASES INHIBITORS FOR THE TREATMENT OF CANCER |
摘要 |
<p>The present invention encompasses compounds of general formula (1) wherein R1 to R3 and X are defined as in claim 1, which are suitable for the treatment of diseases characterized by excessive or abnormal cell proliferation, and the use thereof for preparing a medicament having the above-mentioned properties.</p> |
申请公布号 |
EP2421871(B1) |
申请公布日期 |
2015.09.16 |
申请号 |
EP20100714018 |
申请日期 |
2010.04.21 |
申请人 |
BOEHRINGER INGELHEIM INTERNATIONAL GMBH |
发明人 |
VAN DER VEEN, LARS;IMPAGNATIELLO, MARIA;MCCONNELL, DARRYL;SCHNEIDER, SIEGFRIED;WUNBERG, TOBIAS |
分类号 |
C07D513/04;A61K31/4439;A61P35/00 |
主分类号 |
C07D513/04 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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