发明名称 ANHYDROUS POLYMORPHS OF (2R,3S,4R,5R)-5-(6-(CYCLOPENTYLAMINO)-9H-PURIN-9-YL)-3,4-DIHYDROXYTETRAHYDROFURAN-2-YL) } METHYL NITRATE AND PROCESSES OF PREPARATION THEREOF
摘要 The present invention provides novel anhydrous polymorph forms of 2R,3S,4R,5R)-5-(6-(cyclopentylamino)-9H-purin-9-yl)-3,4-dihydroxytetrahydrofuran-2-yl)methyl nitrate (Compound A). The present invention also provides processes for preparation of the anhydrous polymorphic forms of compound A.
申请公布号 EP2807178(A4) 申请公布日期 2015.09.16
申请号 EP20130741502 申请日期 2013.01.25
申请人 INOTEK PHARMACEUTICALS CORPORATION 发明人 MCVICAR, WILLIAM, K.
分类号 C07H19/167;A61K31/7076;A61P27/02;A61P27/06 主分类号 C07H19/167
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