| 摘要 |
<p>The present invention relates to a first and novel synthetic method of a moracin Y which is contained in mulberry leaves in an infinitesimal amount and exhibits an anticancer activity. The present invention includes a development of a novel synthetic method for efficiently synthesizing the moracin Y through three reaction stages which are a regioselective iodination, a sonogashira coupling, and a desilylation, starting from a 2,4-dihydroxybenzaldehyde which is a cheap compound.</p> |
