发明名称 NOVEL ACETAMIDE DERIVATIVES
摘要 The invention is concerned with a compound of formula (I);;and pharmaceutically acceptable salts thereof wherein R1 to R3, X and Y are as defined as in the description and in the claims. The compound of formula (I) can be used as a medicament.
申请公布号 US2015246906(A1) 申请公布日期 2015.09.03
申请号 US201514712655 申请日期 2015.05.14
申请人 Hoffmann-La Roche Inc. 发明人 BROTHERTON-PLEISS CHRISTINE E.;CHEN ZHI;ERICKSON SHAWN DAVID;QIAN YIMIN
分类号 C07D413/04;C07D207/09;C07D265/30;C07D211/26 主分类号 C07D413/04
代理机构 代理人
主权项 1. A compound of formula (I) wherein: X is —CH2— or oxygen; Y is —(CH2)n—; R1 is phenyl optionally substituted with halogen; R2 is lower alkyl; R3 is trifluoromethyl-phenyl, trifluoromethyl-pyridinyl, trifluoromethyl-pyridazinyl, trifluoromethyl-pyrimidinyl or trifluoromethyl-pyrazinyl; and n is 0 or 1, provided that n is not 0 when X is oxygen; or a pharmaceutically acceptable salt thereof.
地址 Little Falls NJ US