发明名称 1-[2-(2,4-DIMETHYLPHENYLSULFANYL)-PHENYL]PIPERAZINE AS COMPOUND WITH COMBINED SEROTONIN REUPTAKE, 5-HT3 AND 5-HT1A ACTIVITY FOR TREATMENT OF COGNITIVE IMPAIRMENT
摘要 PROBLEM TO BE SOLVED: To provide a compound that is particularly useful for the treatment of cognitive impairment in depressed patients.SOLUTION: This invention provides 1-[2-(2,4-dimethylphenylsulfanyl)-phenyl]piperazine exhibiting strong activity on SERT, 5-HTand 5-HT, which as such can be useful for the treatment of cognitive impairment, in particular, cognitive impairment in depressed patients.
申请公布号 JP2015157872(A) 申请公布日期 2015.09.03
申请号 JP20150118179 申请日期 2015.06.11
申请人 H LUNDBECK AS 发明人 BANG-ANDERSEN BENNY;FALDT ANDRE;MOERK ARNE;LOPEZ DE DIEGO HEIDI;HOLM RENE;STENSBOEL TINE BRYAN;RINGGAARD LONE MUNCH;MEALY MICHAEL J;ROCK MICHAEL HAROLD;BRODERSEN JOERGEN;JOERGENSEN MORTEN;MOORE NICHOLAS
分类号 C07D295/08;A61K31/495;A61P25/00;A61P25/28;A61P43/00 主分类号 C07D295/08
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