发明名称 |
PYRAZOLO[1,5-A]PYRIMIDINE-BASED COMPOUNDS, COMPOSITIONS COMPRISING THEM, AND METHODS OF THEIR USE [15-A] |
摘要 |
<p>Pyrazolo[1,5-a]pyrimidine-based compounds of the formula: are disclosed, wherein R1, R2 and R3 are defined herein. Compositions comprising the compounds and methods of their use to treat, manage and/or prevent diseases and disorders mediated by mediated by adaptor associated kinase 1 activity are also disclosed.</p> |
申请公布号 |
HK1201257(A1) |
申请公布日期 |
2015.08.28 |
申请号 |
HK20150101651 |
申请日期 |
2015.02.13 |
申请人 |
LEXICON PHARMACEUTICALS INC. |
发明人 |
YINGZHI BI;KENNETH GORDON CARSON;GIOVANNI CIANCHETTA;MICHAEL ALAN GREEN;GODWIN KUMI;ALAN MAIN;YULIAN ZHANG;GLENN GREGORY ZIPP |
分类号 |
C07D;A61K;A61P |
主分类号 |
C07D |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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