<p>A method of selectively inhibiting a bromodomain in the presence of other bromodomains comprising introducing a functionally silent mutation into the bromodomain in the presence of other wild type bromodomains and selectively inhibiting the mutated bromodomain.</p>
申请公布号
WO2015079259(A3)
申请公布日期
2015.08.27
申请号
WO2014GB53549
申请日期
2014.11.28
申请人
UNIVERSITY OF DUNDEE;CAMBRIDGE ENTERPRISE LIMITED
发明人
SHIAO, ENRIQUE LIN;BAUD, MATTHIAS GERARD JACKY;CIULLI, ALESSIO;CHAN, KWOK-HO;ZENGERLE, MICHAEL
