发明名称 A RECYCLING PROCESS FOR PREPARING TENOFOVIR ALAFENAMIDE DIASTEREOMERS
摘要 The present invention relates to an efficient and economical process to recycle the undesired diastereomer of Tenofovir alafenamide to desired diastereomer by racemization of the undesired diastereomer followed by separation of the desired diastereomer from the racemic mixture.
申请公布号 WO2015079455(A3) 申请公布日期 2015.08.27
申请号 WO2014IN00734 申请日期 2014.11.27
申请人 LAURUS LABS PRIVATE LIMITED 发明人 THATIPALLY, SURESH;UDUTHA, KUMARA SWAMY;KOTALA, MANI BUSHAN;DAMMALAPATI, VENKATA LAKSHMI NARASIMHA RAO;GORANTLA, SEETA RAMA ANJANEYULU;CHAVA, SATYANARAYANA
分类号 C07D473/34;A61K31/52 主分类号 C07D473/34
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