发明名称 CRYSTALLINE (S)-ISOPROPYL 2-(((S)-(((2R,3R,4R,5R)-5-(2,4-DIOXO-3,4-DIHYDROPYRIMIDIN-1-(2H)-YL)-4-FLUORO-3-HYDROXY-4-METHYLTETRAHYDROFURAN-2-YL)METHOXY)(PHENOXY)PHOSPHORYL)AMINO)PROPANOATE
摘要 <p>Disclosed herein are phosphorus-containing actives, their use as actives for treating diseases, and a stereoselective process for preparing the same. Also disclosed herein are useful synthetic intermediates and processes for preparing the same.</p>
申请公布号 EP2552930(B1) 申请公布日期 2015.08.26
申请号 EP20110714465 申请日期 2011.03.31
申请人 GILEAD PHARMASSET LLC 发明人 ROSS, BRUCE, S.;SOFIA, MICHAEL, JOSEPH;PAMULAPATI, GANAPATI, REDDY;RACHAKONDA, SUGUNA;ZHANG, HAI-REN;CHUN, BYOUNG-KWON;WANG, PEIYUAN
分类号 C07H19/10;A61K31/7072;A61P31/14 主分类号 C07H19/10
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