发明名称 |
CRYSTALLINE (S)-ISOPROPYL 2-(((S)-(((2R,3R,4R,5R)-5-(2,4-DIOXO-3,4-DIHYDROPYRIMIDIN-1-(2H)-YL)-4-FLUORO-3-HYDROXY-4-METHYLTETRAHYDROFURAN-2-YL)METHOXY)(PHENOXY)PHOSPHORYL)AMINO)PROPANOATE |
摘要 |
<p>Disclosed herein are phosphorus-containing actives, their use as actives for treating diseases, and a stereoselective process for preparing the same. Also disclosed herein are useful synthetic intermediates and processes for preparing the same.</p> |
申请公布号 |
EP2552930(B1) |
申请公布日期 |
2015.08.26 |
申请号 |
EP20110714465 |
申请日期 |
2011.03.31 |
申请人 |
GILEAD PHARMASSET LLC |
发明人 |
ROSS, BRUCE, S.;SOFIA, MICHAEL, JOSEPH;PAMULAPATI, GANAPATI, REDDY;RACHAKONDA, SUGUNA;ZHANG, HAI-REN;CHUN, BYOUNG-KWON;WANG, PEIYUAN |
分类号 |
C07H19/10;A61K31/7072;A61P31/14 |
主分类号 |
C07H19/10 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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