Compostos substituidos de enaminocarbolina

摘要

Enaminocarbonyl compounds (I) are new. Enaminocarbonyl compounds of formula (B 1>-C(=O)-C(R 2>)=C(N(R 1>)-A)(D 1>-R 3>)) (I) are new. A : an optionally substituted heterocycle; B 1> : Z-R 4>; Z, T : O, S or optionally substituted N; R 4> : H, 1-6C-alkyl, 1-6C-alkoxy-1-6C-alkyl, 1-6C-alkylthio-1-6C-alkyl, halo-1-6C-alkyl, cyan-1-6C-alkyl, 2-6C-alkenyl, 2-6C-alkynyl, 3-6C-cycloalkyl, 4-10C-dicycloalkyl, tri-1-6C-alkylsilyl, tri-1-6C-alkylsilyl-1-6C-alkyl, hetaryl, hetaryl-1-6C-alkyl, optionally substituted aryl, aryl-1-6C-alkyl or aryl-1-6C-alkoxy-1-6C-alkyl; D 1> : halo, or T-R 5>; R 5> : H, formyl, 1-6C-alkyl, 1-6C-alkoxy-1-6C-alkyl, halo-1-6C-alkoxy-1-6C-alkyl, 1-6C-alkoxy-1-6C-alkoxy-1-6C-alkyl, 1-6C-alkylthio-1-6C-alkyl, 2-6C-alkenyl, 3-6C-cycloalkyl, 2-6C-alkynyl, 1-6C-alkoxycarbonyl, aryl, hetaryl, 1-6C-alkylcarbonyl, aryl-1-6C-alkyl, hetaryl-1-6C-alkyl, halo-1-6C-alkylcarbonyl, arylcarbonyl, 1-6C-alkylsulfonyl, halo-1-6C-alkylsulfonyl, aryl-1-6C-alkyloxy-1-6C-alkyl, aryloxy-1-6C-alkyl, arylsulfonyl or tri-1-6C-alkylsilyl; R 1> : H, 1-6C-alkyl, 2-6C-alkenyl, 1-6C-alkynyl, 3-6C-cycloalkyl, 3-6C-cycloalkyl-1-6C-alkyl, halo-1-6C-alkyl, halo-2-6C-alkenyl, halo-3-6C-cycloalkyl, halo-3-6C-cycloalkyl-1-6C-alkyl, 1-6C-alkoxy or aryl-1-6C-alkyl; R 2> : H or halo; and R 3> : H or 1-6C-alkyl. An independent claim is included for the preparation of (I). ACTIVITY : Insecticide; Arachnicide; Anthelmintic; Nematocide; Acaricide; Fungicide; Antibacterial; Virucide; Herbicide; Antifouling; Plant Growth Regulant. MECHANISM OF ACTION : None given.