发明名称 HETEROAROMATIC AND AROMATIC PIPERAZINYL AZETIDINYL AMIDES AS MONOACYLGLYCEROL LIPASE INHIBITORS
摘要 <p>Disclosed are compounds, compositions and methods for treating diseases, syndromes, conditions and disorders that are affected by the inhibition of MGL, including pain. Such compounds are represented by Formula (I) as follows: wherein Y, r, R2 and Z are defined herein.</p>
申请公布号 HK1170239(A1) 申请公布日期 2015.08.21
申请号 HK20120111003 申请日期 2012.11.01
申请人 JANSSEN PHARMACEUTICA NV 发明人 CHEVALIER, KRISTEN M.;DAX, SCOTT L.;FLORES, CHRISTOPHER M.;LIU, LI;MACIELAG, MARK J.;MC DONNELL, MARK E.;NELEN, MARINA I.;PROUTY, STEPHEN;TODD, MATTHEW;ZHANG, SUI-PO;ZHU, BIN;NULTON, ERICA L.;CLEMENTE, JOSE
分类号 C07D;A61K;A61P 主分类号 C07D
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