发明名称 |
Compostos, composição farmacêutica, métodos de intensificação de eficácia de agente farmacológico e de triagem de compostos para uso como inibidores de mrp e respectivos usos |
摘要 |
<p>5-Quinolinone and Imidazopyrimidine compounds are provided that are useful for inhibiting the efflux of any therapeutic agent that is a MRP1 substrate. Also provided is a method for screening to identify additional MRP1 inhibitors.</p> |
申请公布号 |
BRPI0915467(A2) |
申请公布日期 |
2015.08.18 |
申请号 |
BR2009PI15467 |
申请日期 |
2009.07.10 |
申请人 |
SOUTHERN RESEARCH INSTITUTE |
发明人 |
JOSEPH A. MADDRY;ADAM KEETON;JASON WHITT;GARY PIAZZA |
分类号 |
A01N43/42 |
主分类号 |
A01N43/42 |
代理机构 |
|
代理人 |
|
主权项 |
|
地址 |
|