发明名称 AN EXTENDED RELEASE FORMULATION OF A DIRECT THROMBIN INHIBITOR
摘要 <p>Extended release formulations of 3-fluoro-2-pyridylmethyl-3-(2,2-difluoro-2-(2-pyridyl)ethylamino)-6-chloropyrazin-2-one-1-acetamide (DPOC-4088) that provide for better control of blood plasma levels. The extended release formulations maintain substantially constant plasma levels of the active ingredient for at least about 16 hours and provide for once-daily dosing.</p>
申请公布号 EP2780016(A4) 申请公布日期 2015.08.05
申请号 EP20120848616 申请日期 2012.11.06
申请人 DIAKRON PHARMACEUTICALS, INC. 发明人 RAMAKRISHNAN, SANKAR;VENKATESAN, ELUMALAI;SURYAKUMAR, JAYANTHI;ALLARD, STEPHANE
分类号 A61K31/4965;A61K9/20;A61K31/497;A61P7/02 主分类号 A61K31/4965
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