发明名称 TRIAZOLYL DERIVATIVES AS SYK INHIBITORS
摘要 Provided are triazole derivatives of Formula I which are potent inhibitors of spleen tyrosine kinase and pharmaceutical composition. The triazole derivatives are useful in the treatment and prevention of diseases mediated by said enzyme, such as asthma, COPD, rheumatoid arthritis, and cancer.
申请公布号 EP2900665(A1) 申请公布日期 2015.08.05
申请号 EP20130841430 申请日期 2013.09.24
申请人 MERCK SHARP & DOHME CORP.;MERCK CANADA INC. 发明人 MACHACEK, MICHELLE R.;ROMEO, ERIC T.;KATTAR, SOLOMON D.;CHRISTOPHER, MATTHEW;ALTMAN, MICHAEL D.;NORTHRUP, ALAN B.;ELLIS, JOHN MICHAEL;BOYLE, BRENDAN O';DONOFRIO, ANTHONY;GRIMM, JONATHAN;REUTERSHAN, MICHAEL H.;CHILDERS, KALEEN KONRAD;OTTE, RYAN D.;CASH, BRANDON;DUCHARME, YVES;HAIDLE, ANDREW M.;SPENCER, KERRIE;VITHARANA, DILRUKSHI;WU, LINGYUN;ZHANG, LI;ZHANG, PENG;BEAULIEU, CHRISTIAN;GUAY, DANIEL
分类号 C07D417/12;A61K31/506;A61P11/06;A61P29/00;A61P35/00;C07D239/50;C07D417/14 主分类号 C07D417/12
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