发明名称 NOVEL COMPOUNDS THAT ARE ERK INHIBITORS
摘要 Disclosed are the ERK inhibitors of formula (1.0), having a pyrazolopyridine base structure, and the pharmaceutically acceptable salts thereof. Also disclosed are methods of treating cancer using the compounds of formula (1.0).
申请公布号 EP2900223(A1) 申请公布日期 2015.08.05
申请号 EP20130841687 申请日期 2013.09.26
申请人 MERCK SHARP & DOHME CORP. 发明人 WILSON, KEVIN, J.;WITTER, DAVID, J.;DANIELS, MATTHEW, H.;ANGELES, ANGIE, R.;SILIPHAIVANH, PHIENG;SLOMAN, DAVID;O'BOYLE, BRENDAN;FALCONE, DANIELLE;WHITE, CATHERINE;FERGUSON, RON;ZHOU, WEI;LIPFORD, KATHRYN;MANSOOR, UMAR FARUK;FEVRIER, SALEM;HUANG, XIANHAI;KURUKULASURIYA, RAVI;RICHARD, JUDSON, E.;TANG, SHUYI;BOYCE, CHRISTOPHER;KOZLOWSKI, JOSEPH;BAKSHI, RAMAN KUMAR;KARUNAKARAN, GANESH BABU
分类号 C07D471/04;A61K31/437;A61P35/00 主分类号 C07D471/04
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